Basic Information
ID: ALA4397558
Type: Binding
Description: Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as activation of GalphaS incubated for 5 mins in presence of coelenterazine 400a by BRET assay
Format: BAO_0000219
Organism: Homo sapiens
Target: Beta-1 adrenergic receptor(ALA213)
Document: ALA4396875
Agonist activity at beta1-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as activation of GalphaS incubated for 5 mins in presence of coelenterazine 400a by BRET assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4397558
EC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 415.57 | 4.11 | 4.11 |
| 241.29 | 0.84 | 0.84 |
| 211.26 | 1.13 | 1.13 |
| 437.54 | 3.98 | 3.98 |
| 319.36 | 1.81 | 1.81 |
| 349.38 | 1.51 | 1.51 |
| 467.56 | 3.69 | 3.69 |