Basic Information
ID: ALA4398034
Type: Binding
Description: Agonist activity at recombinant human GABA-A alpha4beta2gamma2S receptor transiently expressed in human tsA201 cells assessed as GABA-induced maximum response incubated for 30 mins and measured up to 90 secs by FMP dye based FLIPR membrane potential blue assay relative to GABA
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4398034
Rmax
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 126.11 | 0.04 | 0.04 |
| 158.18 | 0.35 | 0.35 |
| 160.20 | -0.11 | -0.11 |
| 129.16 | 0.07 | 0.07 |
| 129.16 | 0.07 | 0.07 |
| 174.22 | 0.14 | 0.14 |
| 174.22 | 0.14 | 0.14 |
| 128.13 | -0.54 | -0.54 |
| 174.22 | 0.14 | 0.14 |
| 174.22 | 0.28 | 0.28 |
| 143.15 | -1.25 | -1.25 |
| 160.20 | -0.11 | -0.11 |
| 160.20 | -0.11 | -0.11 |
| 174.22 | 0.28 | 0.28 |
| 174.22 | 0.28 | 0.28 |