Basic Information
ID: ALA4398054
Type: Binding
Description: Inhibition of human GAT3 expressed in Flp-In CHO cells assessed as reduction in [3H]GABA uptake incubated for 3 mins by liquid scintillation counting method
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4398054
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 103.12 | -0.19 | -0.19 |
| 160.20 | -0.11 | -0.11 |
| 129.16 | 0.07 | 0.07 |
| 129.16 | 0.07 | 0.07 |
| 174.22 | 0.14 | 0.14 |
| 174.22 | 0.14 | 0.14 |
| 128.13 | -0.54 | -0.54 |
| 174.22 | 0.14 | 0.14 |
| 174.22 | 0.28 | 0.28 |
| 143.15 | -1.25 | -1.25 |
| 174.22 | 0.28 | 0.28 |