Assay Report Card

Basic Information

ID: ALA4398797

Type: Binding

Description: Inhibition of recombinant human C-terminal His-tagged/N-terminal GST-tagged EGFR (668 to 1210 residues) T790M/L858R/C797S mutant expressed in baculovirus expression system at 100 nM using poly (Glu,Tyr) 4:1 as substrate incubated for 1 hr in presence of ATP by ELISA relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
696.736.866.86