Basic Information
ID: ALA4400461
Type: Binding
Description: Inhibition of human recombinant N-terminal His-tagged and enterokinase cleavage site-fused KLK1 (19 to 262 residues) expressed in baculovirus infected Sf9 insect cells at 10 uM using R110 labelled GSK3162232A as substrate measured at 30 secs interval for 5 mins by FLINT assay relative to control
Format: BAO_0000219
Organism: Homo sapiens
Cell type: Sf9
Target: Kallikrein 1(ALA2319)
Document: ALA4396973
Inhibition of human recombinant N-terminal His-tagged and enterokinase cleavage site-fused KLK1 (19 to 262 residues) expressed in baculovirus infected Sf9 insect cells at 10 uM using R110 labelled GSK3162232A as substrate measured at 30 secs interval for 5 mins by FLINT assay relative to control: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4400461
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 427.67 | ||
| 331.61 | ||
| 423.71 | ||
| 427.67 | ||
| 477.68 | ||
| 423.71 | ||
| 439.71 |