Assay Report Card

Basic Information

ID: ALA4400646

Type: Binding

Description: Inhibition of recombinant mouse 17beta-HSD1 expressed in HEK293 cells at 500 nM using [3H]-E1 as substrate in presence of NAD+ by radio-HPLC analysis relative to control

Organism: Mus musculus

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
573.496.476.47
507.495.715.71
652.397.237.23
503.525.885.88
487.965.955.95
453.525.295.29
523.946.226.22
469.975.815.81
503.525.885.88
487.965.955.95
523.946.226.22
557.496.596.59
469.975.815.81
471.515.435.43