Assay Report Card

Basic Information

ID: ALA4401737

Type: Binding

Description: Inhibition of GAT-1 in rat brain homogenate assessed as decrease in [3H]GABA uptake preincubated for 8 mins followed by [3H]GABA addition and measured after 8 mins by scintillation counting analysis

Organism: Rattus norvegicus

Tissue: Brain

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
375.565.045.04
350.423.173.17