Inhibition of mouse GAT-2 expressed in HEK293 cells assessed as remaining [3H]GABA uptake at 100 uM preincubated for 25 mins followed by [3H]GABA addi...

Basic Information

ID: ALA4401747

Type: Binding

Description: Inhibition of mouse GAT-2 expressed in HEK293 cells assessed as remaining [3H]GABA uptake at 100 uM preincubated for 25 mins followed by [3H]GABA addition and measured after 10 mins by scintillation counting analysis

Format: BAO_0000219

Organism: Mus musculus

Cell type: HEK293

Target:  GABA transporter 3(ALA5205)

Document:  ALA4400545

Inhibition of mouse GAT-2 expressed in HEK293 cells assessed as remaining [3H]GABA uptake at 100 uM preincubated for 25 mins followed by [3H]GABA addition and measured after 10 mins by scintillation counting analysis: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
441.334.294.29
424.883.783.78
424.883.783.78
441.334.294.29