Basic Information
ID: ALA4402772
Type: Binding
Description: Covalent binding affinity to human beta2 adrenoceptor H2.64C mutant expressed in HEK293T cell membranes assessed as covalent blockage of binding site at 5 nM measured within 15 mins by [3H]CGP12177 binding based radioligand depletion assay relative to control
Format: BAO_0000219
Organism: Homo sapiens
Target: Unchecked(ALA612545)
Document: ALA4402511
Covalent binding affinity to human beta2 adrenoceptor H2.64C mutant expressed in HEK293T cell membranes assessed as covalent blockage of binding site at 5 nM measured within 15 mins by [3H]CGP12177 binding based radioligand depletion assay relative to control: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4402772
Activity
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 516.73 | 4.53 | 4.53 |
| 502.70 | 4.14 | 4.14 |