Covalent binding affinity to human beta2 adrenoceptor H2.64C mutant expressed in HEK293T cell membranes assessed as covalent blockage of binding site ...

Basic Information

ID: ALA4402776

Type: Binding

Description: Covalent binding affinity to human beta2 adrenoceptor H2.64C mutant expressed in HEK293T cell membranes assessed as covalent blockage of binding site at 50 nM measured after 30 mins by [3H]CGP12177 binding based radioligand depletion assay relative to control

Format: BAO_0000219

Organism: Homo sapiens

Target:  Unchecked(ALA612545)

Document:  ALA4402511

Covalent binding affinity to human beta2 adrenoceptor H2.64C mutant expressed in HEK293T cell membranes assessed as covalent blockage of binding site at 50 nM measured after 30 mins by [3H]CGP12177 binding based radioligand depletion assay relative to control: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
524.753.573.57