Basic Information
ID: ALA4406027
Type: Binding
Description: Displacement of [3H]CGS21680 from recombinant human A2AAR expressed in HEK293 cell membranes at 10 uM measured after 60 mins by liquid scintillation counting method relative to control
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA4406027
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 451.53 | 2.79 | 2.79 |
| 485.98 | 3.45 | 3.45 |
| 493.54 | 3.13 | 3.13 |
| 498.54 | 1.90 | 1.90 |
| 515.55 | 2.65 | 2.65 |
| 504.02 | 3.82 | 3.82 |
| 511.58 | 2.81 | 2.81 |
| 523.33 | 1.71 | 1.71 |
| 485.52 | 2.64 | 2.64 |
| 533.54 | 2.79 | 2.79 |
| 467.53 | 2.50 | 2.50 |
| 492.00 | 3.51 | 3.51 |
| 538.03 | 3.22 | 3.22 |
| 582.48 | 3.33 | 3.33 |
| 509.99 | 3.65 | 3.65 |
| 527.98 | 3.79 | 3.79 |
| 526.45 | 4.16 | 4.16 |
| 506.03 | 3.82 | 3.82 |
| 483.53 | 2.20 | 2.20 |
| 466.55 | 2.38 | 2.38 |
| 469.52 | 2.93 | 2.93 |
| 497.56 | 2.51 | 2.51 |
| 515.55 | 2.65 | 2.65 |
| 497.56 | 2.51 | 2.51 |