Basic Information
ID: ALA4406540
Type: Binding
Description: Agonist activity at RLuc8-fused human D3R expressed in HEK293 cells co-expressing N-terminal Venus-tagged beta-arrestin2 and GRK3 assessed as induction of beta-arrestin2 recruitment measured after 5 mins in presence of coelenterazine H by BRET assay
Format: BAO_0000219
Organism: Homo sapiens
Cell type: HEK293
Target: Dopamine D3 receptor(ALA234)
Document: ALA4402608
Agonist activity at RLuc8-fused human D3R expressed in HEK293 cells co-expressing N-terminal Venus-tagged beta-arrestin2 and GRK3 assessed as induction of beta-arrestin2 recruitment measured after 5 mins in presence of coelenterazine H by BRET assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4406540
EC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 153.18 | 0.60 | 0.60 |
| 211.33 | 1.58 | 1.58 |
| 379.46 | 3.01 | 3.01 |