Assay Report Card

Basic Information

ID: ALA4413239

Type: Binding

Description: Inhibition of PDK1 in human NCI-H1975 cells assessed as switch of pyruvate metabolism from lactate production to oxidative phosphorylation by measuring decrease in extracellular acidification rate at 1 to 10 uM measured after 4 hrs by XFe24 extracellular flux analyzer based assay

Organism: Homo sapiens

Cell type: NCI-H1975

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
354.443.523.52