Agonist activity at human CB1 receptor expressed in CHO-RD-HGA16 cells co-expressing Galpha16 assessed as suppression stimulation of calcium mobilizat...

Basic Information

ID: ALA4416379

Type: Functional

Description: Agonist activity at human CB1 receptor expressed in CHO-RD-HGA16 cells co-expressing Galpha16 assessed as suppression stimulation of calcium mobilization incubated for 45 mins by Calcium 5 dye based FLIPR assay relative to CP55,940

Format: BAO_0000219

Organism: Homo sapiens

Target:  Cannabinoid CB1 receptor(ALA218)

Document:  ALA4414612

Agonist activity at human CB1 receptor expressed in CHO-RD-HGA16 cells co-expressing Galpha16 assessed as suppression stimulation of calcium mobilization incubated for 45 mins by Calcium 5 dye based FLIPR assay relative to CP55,940: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
392.895.655.65
342.856.026.02
358.855.725.72
323.785.055.05
286.764.024.02
371.895.785.78
397.717.027.02
346.815.855.85
323.785.055.05
363.276.376.37
286.764.024.02
370.865.925.92
397.717.027.02
329.834.134.13
358.855.725.72
328.825.715.71
328.825.715.71
323.785.055.05
422.925.655.65
328.825.715.71
363.276.376.37
406.925.125.12
363.276.376.37
346.815.855.85
386.865.505.50
323.785.055.05
329.815.115.11
329.815.115.11
358.855.725.72
364.805.995.99
329.815.115.11