Agonist activity at human CB2 receptor expressed in CHO cells co-expressing Galpha16 assessed as increase in calcium mobilization at 10 uM measured at...

Basic Information

ID: ALA4416380

Type: Functional

Description: Agonist activity at human CB2 receptor expressed in CHO cells co-expressing Galpha16 assessed as increase in calcium mobilization at 10 uM measured at 1 sec interval for 90 secs by calcium-5 dye based FLIPR assay relative to CP55,940

Format: BAO_0000219

Organism: Homo sapiens

Cell type: CHO

Target:  Cannabinoid CB2 receptor(ALA253)

Document:  ALA4414612

Agonist activity at human CB2 receptor expressed in CHO cells co-expressing Galpha16 assessed as increase in calcium mobilization at 10 uM measured at 1 sec interval for 90 secs by calcium-5 dye based FLIPR assay relative to CP55,940: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
392.895.655.65
342.856.026.02
358.855.725.72
323.785.055.05
286.764.024.02
371.895.785.78
397.717.027.02
346.815.855.85
323.785.055.05
363.276.376.37
286.764.024.02
370.865.925.92
397.717.027.02
329.834.134.13
358.855.725.72
328.825.715.71
328.825.715.71
323.785.055.05
422.925.655.65
328.825.715.71
363.276.376.37
406.925.125.12
363.276.376.37
346.815.855.85
386.865.505.50
323.785.055.05
329.815.115.11
329.815.115.11
358.855.725.72
364.805.995.99
329.815.115.11