Basic Information
ID: ALA4417505
Type: Binding
Description: Inhibition of N-terminal GST-tagged human EGFR cytoplasmic domain (669-1210 AA) expressed in baculovirus at 10 uM using FAM-labelled peptide as substrate pre-incubated for 10 mins followed by substrate addition by mobility shift assay relative to control
Format: BAO_0000019
Organism: Homo sapiens
Target: Epidermal growth factor receptor erbB1(ALA203)
Document: ALA4414679
Inhibition of N-terminal GST-tagged human EGFR cytoplasmic domain (669-1210 AA) expressed in baculovirus at 10 uM using FAM-labelled peptide as substrate pre-incubated for 10 mins followed by substrate addition by mobility shift assay relative to control: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4417505
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 483.15 | 5.94 | 5.94 |
| 434.28 | 5.19 | 5.19 |
| 463.42 | 4.91 | 4.91 |
| 393.45 | 4.50 | 4.50 |
| 406.25 | 5.62 | 5.62 |
| 402.29 | 5.79 | 5.79 |
| 418.28 | 5.49 | 5.49 |
| 463.42 | 4.91 | 4.91 |
| 430.34 | 6.47 | 6.47 |
| 521.32 | 4.49 | 4.49 |
| 521.32 | 4.49 | 4.49 |
| 402.29 | 5.73 | 5.73 |
| 472.25 | 6.20 | 6.20 |
| 426.67 | 5.96 | 5.96 |
| 409.45 | 4.20 | 4.20 |
| 421.50 | 5.18 | 5.18 |
| 422.25 | 5.32 | 5.32 |
| 406.25 | 5.62 | 5.62 |
| 393.45 | 4.44 | 4.44 |
| 421.50 | 5.18 | 5.18 |
| 434.28 | 5.19 | 5.19 |
| 417.83 | 4.67 | 4.67 |
| 483.15 | 5.94 | 5.94 |
| 425.45 | 3.90 | 3.90 |
| 474.32 | 4.65 | 4.65 |
| 397.41 | 4.33 | 4.33 |
| 425.45 | 3.90 | 3.90 |
| 397.41 | 4.33 | 4.33 |
| 393.45 | 4.44 | 4.44 |
| 430.34 | 6.47 | 6.47 |
| 474.32 | 4.65 | 4.65 |
| 413.41 | 4.03 | 4.03 |
| 472.25 | 6.20 | 6.20 |