Basic Information
ID: ALA4418371
Type: Binding
Description: Inhibition of recombinant GST-tagged human PASK kinase domain (879 to 1323 residues) expressed in baculovirus expression system using Ulight peptide as substrate incubated for 2 hrs under dark condition by TR-FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4418371
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 242.24 | 1.09 | 1.09 |
| 387.23 | 4.07 | 4.07 |
| 370.77 | 3.55 | 3.55 |
| 366.76 | 3.13 | 3.13 |
| 352.78 | 3.41 | 3.41 |
| 346.35 | 2.40 | 2.40 |
| 329.32 | 2.02 | 2.02 |
| 266.26 | 1.27 | 1.27 |
| 280.29 | 1.52 | 1.52 |
| 281.28 | 0.92 | 0.92 |
| 310.28 | -0.28 | -0.28 |
| 397.23 | 3.93 | 3.93 |
| 398.21 | 3.33 | 3.33 |
| 362.78 | 3.28 | 3.28 |
| 363.77 | 2.68 | 2.68 |
| 295.31 | 1.48 | 1.48 |
| 284.28 | 1.16 | 1.16 |
| 270.25 | 0.86 | 0.86 |
| 360.37 | 2.45 | 2.45 |
| 332.36 | 2.68 | 2.68 |
| 346.33 | 2.77 | 2.77 |
| 374.38 | 3.26 | 3.26 |
| 363.77 | 2.68 | 2.68 |
| 343.35 | 2.33 | 2.33 |
| 296.25 | -0.55 | -0.55 |
| 390.83 | 3.77 | 3.77 |
| 256.26 | 1.40 | 1.40 |
| 347.33 | 1.92 | 1.92 |
| 333.31 | 1.88 | 1.88 |
| 363.77 | 2.68 | 2.68 |
| 347.31 | 2.16 | 2.16 |
| 329.32 | 2.02 | 2.02 |
| 390.83 | 3.77 | 3.77 |
| 267.25 | 0.66 | 0.66 |
| 362.78 | 3.28 | 3.28 |
| 343.35 | 1.95 | 1.95 |
| 344.34 | 1.34 | 1.34 |