Assay Report Card

Basic Information

ID: ALA4418544

Type: Binding

Description: Inhibition of TMPRSS4 serine protease domain (Val205 to Leu437 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) at 30 uM using Z-Phe-Arg7-amido-4-methylcoumarin hydrochloride substrate measured at 5 mins interval for 150 mins by fluorescence based assay relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
349.234.684.68
254.702.752.75
248.672.692.69
383.685.345.34
272.693.173.17
315.684.324.32
247.683.303.30
315.684.324.32
275.743.913.91
272.693.173.17
316.574.604.60
329.704.634.63
350.124.974.97
333.674.464.46
394.575.085.08
333.674.464.46
350.124.974.97
340.694.194.19
345.704.334.33
351.025.265.26
363.264.994.99
367.224.824.82
428.135.445.44
379.264.694.69
418.125.995.99
394.234.594.59
425.715.565.56
473.807.217.21
397.705.015.01
383.685.345.34
383.685.345.34
394.575.085.08
413.705.345.34
462.576.106.10
384.664.734.73
400.285.235.23
273.682.562.56
316.673.713.71
283.113.353.35
283.113.353.35
249.662.092.09
298.733.853.85
383.685.345.34
383.685.345.34
374.244.554.55
392.263.783.78
277.712.702.70
268.733.063.06
322.693.773.77
397.705.645.64
331.783.823.82
351.114.374.37
320.633.253.25
283.113.353.35
360.684.224.22
256.711.881.88
394.575.085.08
364.254.264.26
495.757.287.28
330.804.424.42
323.683.173.17
417.235.705.70
268.733.063.06
366.565.575.57
307.143.823.82
251.672.032.03
418.125.995.99
406.284.644.64
418.125.995.99
399.295.845.84
381.893.363.36
308.793.633.63
283.113.353.35
252.661.721.72
282.753.373.37