Assay Report Card

Basic Information

ID: ALA4419742

Type: Binding

Description: Inhibition of GST-tagged human DBL RhoGEF DH-PH module expressed in mouse NIH/3T3 cells assessed as reduction in human full length RhoA (1 to 193 residues) interaction with DBL RhoGEF at 10 to 50 uM incubated for 1 hr by Western blot analysis based His-RhoA pull-down assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
384.444.044.04