Basic Information
ID: ALA4420050
Type: Functional
Description: Antagonist activity at recombinant human MrgprX4 expressed in HEK293 cells assessed as blockade of bilirubin-induced inositol phosphate accumulation incubated for 1 hr at at 37 degC followed by incubation for 30 mins at room temperature before bilirubin addition by HTRF assay relative to control
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA4420050
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 287.75 | 3.35 | 3.35 |
| 407.82 | 4.84 | 4.84 |
| 457.33 | 5.47 | 5.47 |
| 348.84 | 4.95 | 4.95 |