Assay Report Card

Basic Information

ID: ALA4424780

Type: Binding

Description: Inhibition of human C-terminal FLAG-tagged KDM5A (1 to 1090 residues) expressed in baculovirus infected Sf9 insect cells at 1 uM using H3(1-21)K4(Me3)-GGK(Biotin)/2-OG as substrate measured after 1 hr by Alphalisa assay relative to control

Organism: Homo sapiens

Cell type: Sf9

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
288.391.971.97
384.483.083.08
278.312.682.68
321.422.412.41
405.554.704.70
375.472.152.15