Assay Report Card

Basic Information

ID: ALA4424791

Type: Binding

Description: Inhibition of human N-terminal His-tagged KDM4A (1 to 350 residues) expressed in Escherichia coli at 25 uM using H3(21-44)-K36(Me3)-GK(Biotin)/2-OG as substrate measured after 1 hr by Alphalisa assay relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
288.391.971.97
278.312.682.68
405.554.704.70
419.574.744.74