Basic Information
ID: ALA4425808
Type: Binding
Description: Inhibition of human recombinant GST-tagged DDR1 (440 to 876 residues) expressed in baculovirus infected Sf9 insect cells using fluorescein-poly GAT as substrate preincubated for 1 hr measured after 1 hr in presence of ATP by TR-FRET LanthaScreen assay
Format: BAO_0000219
Organism: Homo sapiens
Cell type: Sf9
Target: Epithelial discoidin domain-containing receptor 1(ALA5319)
Document: ALA4425102
Inhibition of human recombinant GST-tagged DDR1 (440 to 876 residues) expressed in baculovirus infected Sf9 insect cells using fluorescein-poly GAT as substrate preincubated for 1 hr measured after 1 hr in presence of ATP by TR-FRET LanthaScreen assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4425808
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 524.59 | 4.62 | 4.62 |
| 510.56 | 4.06 | 4.06 |
| 538.62 | 5.01 | 5.01 |
| 524.59 | 4.62 | 4.62 |
| 492.51 | 5.37 | 5.37 |
| 552.65 | 5.25 | 5.25 |
| 508.59 | 5.27 | 5.27 |
| 509.58 | 4.66 | 4.66 |
| 492.51 | 5.37 | 5.37 |
| 538.62 | 5.01 | 5.01 |
| 552.65 | 5.25 | 5.25 |