Basic Information
ID: ALA4426323
Type: Binding
Description: Displacement of [125I]-ET-1 from human ETA receptor expressed in CHO cell membranes after 2 hrs by scintillation counting
Organism: Homo sapiens
Cell type: CHO
Activity Charts
Bioactivity
Activity Types for Assay ALA4426323
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 410.43 | 2.92 | 2.92 |
| 450.51 | 5.59 | 5.59 |
| 432.48 | 2.44 | 2.44 |
| 378.43 | 3.52 | 3.52 |
| 659.81 | 5.28 | 5.28 |
| 424.44 | 2.71 | 2.71 |
| 588.28 | 3.57 | 3.57 |
| 517.48 | 5.05 | 5.05 |
| 546.20 | 2.53 | 2.53 |
| 469.52 | 2.50 | 2.50 |
| 511.03 | 3.42 | 3.42 |
| 522.61 | 2.90 | 2.90 |
| 674.74 | 4.07 | 4.07 |
| 529.80 | 3.07 | 3.07 |
| 569.51 | 3.92 | 3.92 |
| 525.06 | 3.81 | 3.81 |
| 618.26 | 2.64 | 2.64 |
| 626.70 | 5.02 | 5.02 |
| 555.48 | 3.53 | 3.53 |
| 522.61 | 2.90 | 2.90 |
| 553.44 | 3.21 | 3.21 |
| 541.06 | 3.43 | 3.43 |
| 495.00 | 5.09 | 5.09 |
| 539.41 | 2.82 | 2.82 |
| 527.43 | 2.75 | 2.75 |
| 527.03 | 3.04 | 3.04 |
| 656.74 | 4.18 | 4.18 |
| 571.48 | 2.77 | 2.77 |
| 510.61 | 4.82 | 4.82 |
| 541.45 | 3.14 | 3.14 |
| 482.98 | 2.64 | 2.64 |
| 649.71 | 5.11 | 5.11 |
| 555.41 | 2.94 | 2.94 |
| 620.09 | 4.56 | 4.56 |
| 497.00 | 3.03 | 3.03 |
| 568.45 | 4.87 | 4.87 |
| 545.98 | 1.95 | 1.95 |