Agonist activity at GST-tagged FXR-LBD (unknown origin) assessed as biotin-labeled SRC-1 recruitment at 5 uM after 30 mins by Alpha Screen assay relat...

Basic Information

ID: ALA4433551

Type: Binding

Description: Agonist activity at GST-tagged FXR-LBD (unknown origin) assessed as biotin-labeled SRC-1 recruitment at 5 uM after 30 mins by Alpha Screen assay relative to 6-ECDCA

Format: BAO_0000357

Organism: Homo sapiens

Target:  Bile acid receptor FXR(ALA2047)

Document:  ALA4433207

Agonist activity at GST-tagged FXR-LBD (unknown origin) assessed as biotin-labeled SRC-1 recruitment at 5 uM after 30 mins by Alpha Screen assay relative to 6-ECDCA: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
542.858.878.87
392.584.484.48
392.285.845.84
482.367.727.72
387.276.226.22
392.285.845.84
362.266.356.35
498.417.427.42
526.427.727.72
440.355.755.75
493.397.807.80
406.276.056.05
387.276.226.22
526.427.727.72
420.296.146.14
498.417.427.42
496.397.807.80
493.397.807.80
468.387.517.51
512.397.637.63
420.296.146.14
512.397.637.63
406.276.056.05