Assay Report Card

ID: ALA4478073

Type: Binding

Description: Binding affinity to human NPY Y4 receptor expressed in CHO cells co-expressing Gqi5-mtAEQ assessed as slow dissociation half life t1/2(2) at 1.5 uM incubated for 2 hrs in presence of 200-fold excess of N'-[(2S)-2-[[(2S)-5-[[N'-(4-aminobutylcarbamoyl)carbamimidoyl]amino]-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-5-guanidino-pentanoyl]amino]-4-methyl-pentanoyl]amino]pentanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]-N-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-5-guanidino-pentanoyl]amino]-4-methyl-pentanoyl]amino]-5-guanidino-pentanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]octanediamide by liquid scintillation counting

Organism: Homo sapiens

Cell type: CHO