Basic Information
ID: ALA4478089
Type: Binding
Description: Antagonist activity at recombinant human TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced intracellular calcium accumulation preincubated for 5 mins followed by capsaicin addition by Fluo-4-AM probe-based spectrofluorimetric assay
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA4478089
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 588.66 | 4.37 | 4.37 |
| 564.68 | 6.44 | 6.44 |
| 600.66 | 6.71 | 6.71 |
| 633.57 | 7.74 | 7.74 |