Assay Report Card

Basic Information

ID: ALA4478096

Type: Binding

Description: Antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced intracellular calcium accumulation up to 10 uM preincubated for 5 mins followed by LPC addition by Fluo-4-AM probe-based spectrofluorimetric assay

Organism: Rattus norvegicus

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
588.664.374.37
564.686.446.44
600.666.716.71
633.577.747.74