Basic Information
ID: ALA4605123
Type: Binding
Description: Inhibition of recombinant human full-length N-terminal GST-tagged CDK9/cyclinK expressed in baculovirus infected Sf9 insect cells using PDKtide as substrate measured after 120 mins by ADP-glo assay
Format: BAO_0000219
Organism: Homo sapiens
Cell type: Sf9
Target: CDK9/Cyclin K(ALA3038475)
Document: ALA4602695
Inhibition of recombinant human full-length N-terminal GST-tagged CDK9/cyclinK expressed in baculovirus infected Sf9 insect cells using PDKtide as substrate measured after 120 mins by ADP-glo assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4605123
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 447.54 | 2.97 | 2.97 |
| 506.61 | 4.94 | 4.94 |
| 513.09 | 4.88 | 4.88 |
| 425.92 | 3.77 | 3.77 |
| 311.78 | 4.32 | 4.32 |
| 396.88 | 4.16 | 4.16 |
| 274.76 | 3.76 | 3.76 |
| 310.79 | 4.93 | 4.93 |
| 395.90 | 3.76 | 3.76 |
| 399.89 | 3.23 | 3.23 |
| 423.95 | 4.46 | 4.46 |
| 495.03 | 5.98 | 5.98 |
| 408.94 | 4.68 | 4.68 |
| 311.78 | 4.32 | 4.32 |
| 479.89 | 4.66 | 4.66 |
| 439.95 | 3.64 | 3.64 |
| 453.98 | 3.68 | 3.68 |
| 423.95 | 4.33 | 4.33 |
| 325.80 | 4.19 | 4.19 |
| 324.82 | 5.23 | 5.23 |
| 477.92 | 4.65 | 4.65 |
| 409.93 | 4.07 | 4.07 |
| 316.84 | 4.93 | 4.93 |
| 314.78 | 4.39 | 4.39 |
| 413.89 | 3.90 | 3.90 |
| 441.94 | 3.81 | 3.81 |
| 422.96 | 5.07 | 5.07 |
| 395.89 | 4.76 | 4.76 |
| 395.90 | 3.73 | 3.73 |
| 452.01 | 5.06 | 5.06 |
| 338.84 | 4.84 | 4.84 |
| 311.78 | 4.32 | 4.32 |
| 409.93 | 4.07 | 4.07 |
| 341.80 | 4.33 | 4.33 |
| 441.94 | 3.81 | 3.81 |
| 409.93 | 3.63 | 3.63 |
| 409.93 | 4.07 | 4.07 |
| 393.92 | 5.92 | 5.92 |
| 463.89 | 4.78 | 4.78 |
| 437.98 | 4.89 | 4.89 |
| 339.83 | 4.23 | 4.23 |
| 437.98 | 4.89 | 4.89 |
| 481.89 | 4.92 | 4.92 |
| 346.22 | 4.97 | 4.97 |
| 422.96 | 5.07 | 5.07 |
| 425.92 | 3.77 | 3.77 |
| 394.91 | 5.31 | 5.31 |
| 479.89 | 4.66 | 4.66 |
| 439.95 | 3.64 | 3.64 |
| 439.95 | 3.64 | 3.64 |
| 423.95 | 3.94 | 3.94 |
| 423.95 | 3.68 | 3.68 |
| 413.89 | 3.90 | 3.90 |
| 324.82 | 4.79 | 4.79 |
| 437.98 | 4.89 | 4.89 |
| 437.98 | 4.69 | 4.69 |
| 452.95 | 3.72 | 3.72 |
| 339.83 | 4.23 | 4.23 |
| 413.89 | 3.90 | 3.90 |
| 427.92 | 3.77 | 3.77 |