ID: ALA4605235
Type: Binding
Description: Antagonist activity at muscarinic M3 receptor (unknown origin) expressed in HEK293 cells coexpressing EA tagged beta-arrestin2 assessed as inhibition of carbachol-induced beta-arrestin2 recruitment preincubated for 30 mins followed by carbachol addition and measured after 90 mins by PathHunter assay
Organism: Homo sapiens
Cell type: HEK293
Bioactivity
Activity Types for Assay ALA4605235
EC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
426.56 | 3.96 | 3.96 |
452.89 | 5.07 | 5.07 |
380.82 | 4.83 | 4.83 |
472.43 | 2.35 | 2.35 |
392.83 | 4.93 | 4.93 |
362.83 | 4.69 | 4.69 |
434.90 | 4.93 | 4.93 |
374.84 | 4.79 | 4.79 |