Basic Information
ID: ALA4612475
Type: Binding
Description: Displacement of APC-labeled biotinylated-avidin from Euphorium-chelated recombinant human BRD4 bromodomain 1 expressed in Escherichia coli preincubated for 15 mins followed by APC-labeled biotinylated-avidin addition and measured after 1 hr under dark condition by TR-FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4612475
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 457.00 | 5.53 | 5.53 |
| 538.63 | 4.46 | 4.46 |
| 464.52 | 4.05 | 4.05 |
| 530.63 | 5.68 | 5.68 |
| 464.52 | 4.05 | 4.05 |
| 440.53 | 2.90 | 2.90 |
| 478.55 | 4.36 | 4.36 |
| 465.51 | 3.44 | 3.44 |
| 536.66 | 5.89 | 5.89 |
| 478.55 | 4.36 | 4.36 |
| 502.58 | 5.05 | 5.05 |
| 478.55 | 4.44 | 4.44 |
| 492.58 | 4.66 | 4.66 |
| 503.61 | 5.32 | 5.32 |
| 479.54 | 3.83 | 3.83 |
| 488.61 | 4.92 | 4.92 |
| 479.54 | 3.83 | 3.83 |
| 464.52 | 4.05 | 4.05 |
| 566.69 | 5.24 | 5.24 |
| 474.59 | 4.52 | 4.52 |
| 552.66 | 4.85 | 4.85 |
| 460.51 | 3.91 | 3.91 |