Assay Report Card

Basic Information

ID: ALA4612762

Type: Binding

Description: Inhibition of recombinant human full-length N-terminal GST-tagged CDK2/cyclinA1 expressed in baculovirus infected Sf9 insect cells using FRET-labeled Ser/Thr 12 as substrate measured after 1 hr by Z'-lyte assay

Organism: Homo sapiens

Cell type: Sf9

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
380.543.663.66
522.684.564.56
593.706.586.58
523.664.994.99
525.705.565.56
561.685.815.81
507.665.065.06
539.735.875.87
479.634.674.67
548.625.095.09
434.594.084.08
442.575.105.10
486.664.504.50
539.735.955.95
543.695.705.70
539.735.955.95
553.715.345.34
526.694.964.96
555.105.555.55
525.705.565.56
511.726.686.68
541.704.584.58
526.694.964.96