Assay Report Card

Basic Information

ID: ALA4612763

Type: Binding

Description: Inhibition of recombinant human full-length His-tagged CDK7/Cyclin H/MNAT1 expressed in baculovirus infection system using Cdk7/9tide as substrate measured after 1 hr by Alexa Fluor 647 ADP Tracer-based Adapta assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
380.543.663.66
522.684.564.56
593.706.586.58
523.664.994.99
525.705.565.56
561.685.815.81
507.665.065.06
539.735.875.87
479.634.674.67
548.625.095.09
434.594.084.08
442.575.105.10
486.664.504.50
539.735.955.95
543.695.705.70
539.735.955.95
553.715.345.34
526.694.964.96
555.105.555.55
525.705.565.56
511.726.686.68
541.704.584.58
526.694.964.96