Assay Report Card

Basic Information

ID: ALA4612764

Type: Binding

Description: Inhibition of recombinant human full-length His-tagged CDK9/Cyclin T1 expressed in baculovirus infection system using Cdk7/9tide as substrate measured after 1 hr in presence of Alexa Fluor 647 ADP Tracer-based Adapta assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
380.543.663.66
522.684.564.56
593.706.586.58
523.664.994.99
525.705.565.56
561.685.815.81
507.665.065.06
539.735.875.87
479.634.674.67
548.625.095.09
434.594.084.08
442.575.105.10
486.664.504.50
539.735.955.95
543.695.705.70
539.735.955.95
553.715.345.34
526.694.964.96
555.105.555.55
525.705.565.56
511.726.686.68
541.704.584.58
526.694.964.96