Basic Information
ID: ALA4612790
Type: Binding
Description: Inhibition of CDK12 C1039S mutant in human HAP1 cells assessed as reduction in RNA Polymerase 2 CTD phosphorylation at Ser5 residues at 40 to 200 nM measured after 6 hrs by Western blot analysis
Organism: Homo sapiens
Cell type: HAP1
Activity Charts
Bioactivity
Activity Types for Assay ALA4612790
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 525.70 | 5.56 | 5.56 |