Assay Report Card

Basic Information

ID: ALA4612792

Type: Binding

Description: Inhibition of CDK12 C1039S mutant in human HAP1 cells assessed as reduction in RNA Polymerase 2 expression at 40 to 200 nM measured after 6 hrs by Western blot analysis

Organism: Homo sapiens

Cell type: HAP1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
525.705.565.56