Assay Report Card

Basic Information

ID: ALA4615928

Type: Binding

Description: Inhibition of recombinant full length human N-terminal GST-tagged GSK3beta (1 to 420 end residues) expressed in baculovirus expression system using unphosphorylated peptide as substrate incubated enzyme-substrate mixture for 90 mins in presence of ATP by LANCE assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
466.544.354.35
428.483.603.60
394.483.573.57
391.402.432.43
343.333.033.03
357.363.423.42
357.363.423.42
357.363.273.27
371.393.663.66
357.363.423.42
380.452.932.93
336.402.782.78
366.422.272.27
371.393.663.66
366.422.272.27
380.452.932.93
405.432.822.82