Basic Information
ID: ALA4620602
Type: Binding
Description: Inhibition of human recombinant Haspin (470 to 798 residues) expressed in bacteria assessed as residual activity at 1 uM using Histone H3 and ARTKQTARKSTGGKAPRKQLA as substrate in presence of ATP incubated for 50 mins by ADP-GloTM assay relative to control
Format: BAO_0000019
Organism: Homo sapiens
Target: Serine/threonine-protein kinase haspin(ALA1075163)
Document: ALA4619742
Inhibition of human recombinant Haspin (470 to 798 residues) expressed in bacteria assessed as residual activity at 1 uM using Histone H3 and ARTKQTARKSTGGKAPRKQLA as substrate in presence of ATP incubated for 50 mins by ADP-GloTM assay relative to control: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4620602
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 146.15 | 1.38 | 1.38 |
| 320.35 | 3.40 | 3.40 |
| 304.35 | 3.78 | 3.78 |
| 276.30 | 3.22 | 3.22 |
| 290.32 | 3.48 | 3.48 |
| 292.36 | 3.93 | 3.93 |
| 304.35 | 3.78 | 3.78 |
| 290.32 | 3.39 | 3.39 |
| 260.30 | 3.39 | 3.39 |
| 278.27 | 2.88 | 2.88 |
| 334.38 | 3.79 | 3.79 |
| 274.32 | 3.78 | 3.78 |
| 304.31 | 3.11 | 3.11 |