Assay Report Card

Basic Information

ID: ALA4621236

Type: ADME

Description: Inhibition of recombinant human His-tagged MMP3 catalytic domain (Pro19 to Glu271 residues) expressed in Escherichia coli at 100 uM using 5-FAM/QXL520-labelled FRET peptide as substrate preincubated for 10 to 15 mins followed by substrate addition and measured every minute for 1 hr by FRET assay relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
249.291.451.45
276.142.562.56