Assay Report Card

Basic Information

ID: ALA4622279

Type: Binding

Description: Antagonist activity at human VDR expressed in HEK293 EBNA cells co-expressing CYP24A1 promoter region assessed as reduction in 1,25D3-induced receptor activation at 0.1 to 1000 nM incubated for 18 hrs by luciferase reporter gene assay relative to control

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
510.725.585.58