Assay Report Card

Basic Information

ID: ALA4626993

Type: Binding

Description: Selectivity index, difference between pIC50 for N-terminal His6-tagged human BRD2 BD1 (1 to 473 residues)/ BD2 Y386A mutant expressed in Escherichia coli to pIC50 for N-terminal His6-tagged human BRD2 BD2 (1 to 473 residues)/BD1 Y113A mutant expressed in Escherichia coli

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
415.454.164.16
442.525.625.62
511.635.605.60