Basic Information
ID: ALA4630174
Type: Binding
Description: Inhibition of recombinant N-terminal His-tagged LSD1 (unknown origin) expressed in Escherichia coli expression system using ART-K(Me1)-QTARKSTGGKAPRKQLAGGK(Biotin) as substrate incubated for 60 mins by TR-FRET assay
Format: BAO_0000019
Organism: Homo sapiens
Target: Lysine-specific histone demethylase 1(ALA6136)
Document: ALA4627402
Inhibition of recombinant N-terminal His-tagged LSD1 (unknown origin) expressed in Escherichia coli expression system using ART-K(Me1)-QTARKSTGGKAPRKQLAGGK(Biotin) as substrate incubated for 60 mins by TR-FRET assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4630174
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 133.19 | 1.50 | 1.50 |
| 364.49 | 3.74 | 3.74 |
| 159.23 | 2.05 | 2.05 |
| 159.23 | 2.05 | 2.05 |
| 360.52 | 2.88 | 2.88 |
| 314.47 | 2.91 | 2.91 |
| 185.27 | 2.36 | 2.36 |
| 338.50 | 3.32 | 3.32 |
| 328.50 | 3.35 | 3.35 |
| 354.54 | 3.70 | 3.70 |
| 253.35 | 2.99 | 2.99 |
| 137.23 | 1.83 | 1.83 |
| 356.51 | 3.83 | 3.83 |
| 270.42 | 3.07 | 3.07 |
| 187.29 | 2.83 | 2.83 |
| 324.47 | 3.47 | 3.47 |
| 256.39 | 2.68 | 2.68 |
| 173.26 | 2.44 | 2.44 |
| 271.40 | 3.37 | 3.37 |
| 270.42 | 3.34 | 3.34 |
| 342.48 | 3.44 | 3.44 |
| 270.38 | 2.35 | 2.35 |
| 173.26 | 2.44 | 2.44 |
| 256.39 | 2.82 | 2.82 |
| 326.48 | 2.91 | 2.91 |
| 314.47 | 2.96 | 2.96 |
| 282.43 | 3.21 | 3.21 |
| 228.34 | 2.04 | 2.04 |
| 346.47 | 4.19 | 4.19 |
| 312.46 | 3.52 | 3.52 |