Assay Report Card

Basic Information

ID: ALA4630226

Type: Functional

Description: Antagonist activity at N-terminal HA-tagged and C-terminal FLAG-tagged human MC4R expressed in HEK293 cells assessed as reduction in alpha-MSH-induced cAMP accumulation at 100 uM incubated for 3 hrs by luciferase reporter gene assay

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
2915.51
3795.71