Assay Report Card

Basic Information

ID: ALA4630482

Type: Binding

Description: Antagonist activity at human Gi/G0-coupled CXCR4 assessed as inhibition of CXCL12-induced beta arrestin2 recruitment at 500 nM preincubated for 30 mins followed by CXCL12 stimulation and measured after 90 to 180 mins by pathhunter assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
500.433.753.75