Basic Information
ID: ALA4667412
Type: Binding
Description: Selectivity index, ratio of EC50 for RORalpha (unknown origin) to EC50 for His-tagged RORgammat (T259 to K518 residues) (unknown origin) using PGC1alpha as co-activator incubated for 1 hr by AlphaScreen and cofactor recruitment assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4667412
Ratio EC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 427.37 | 4.21 | 4.21 |
| 588.52 | 4.73 | 4.73 |
| 562.40 | 5.09 | 5.09 |
| 616.57 | 5.54 | 5.54 |
| 574.49 | 4.51 | 4.51 |
| 562.44 | 5.77 | 5.77 |
| 519.37 | 6.23 | 6.23 |
| 602.54 | 5.33 | 5.33 |
| 563.38 | 5.69 | 5.69 |
| 604.48 | 6.16 | 6.16 |
| 549.40 | 5.59 | 5.59 |
| 533.40 | 6.62 | 6.62 |
| 613.57 | 6.21 | 6.21 |
| 584.53 | 6.00 | 6.00 |
| 642.61 | 6.72 | 6.72 |
| 577.45 | 6.23 | 6.23 |
| 576.42 | 5.35 | 5.35 |
| 585.51 | 5.39 | 5.39 |
| 590.45 | 5.60 | 5.60 |
| 585.51 | 5.39 | 5.39 |
| 507.53 | 4.04 | 4.04 |
| 563.42 | 6.25 | 6.25 |
| 628.46 | 5.22 | 5.22 |
| 588.52 | 4.73 | 4.73 |
| 558.41 | 6.37 | 6.37 |
| 614.55 | 5.91 | 5.91 |
| 563.43 | 6.25 | 6.25 |
| 585.51 | 5.39 | 5.39 |