Assay Report Card

Basic Information

ID: ALA4667970

Type: Binding

Description: Inhibition of recombinant Trypanosoma brucei rhodesain expressed in Pichia pastoris at 10 uM using Z-FR-AMC as substrate and measured at 12 sec interval for 5 mins without preincubation by fluorimetric analysis relative to control

Organism: Trypanosoma brucei

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
270.334.904.90
367.283.703.70
438.904.044.04
395.893.283.28
403.924.794.79
341.724.164.16
357.414.884.88
326.404.994.99
268.144.114.11
362.444.504.50
293.323.763.76
400.464.424.42
489.525.365.36
456.644.454.45