Assay Report Card

Basic Information

ID: ALA4670360

Type: Functional

Description: Partial agonist activity at SNAP-tagged human GHSR expressed in HEK293 cells assessed as stimulation of ghrelin-induced increase in IP1 accumulation at 10^-5 M measured after 30 mins by IP1-d2 derivative based HTRF assay relative to ghrelin

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
536.643.753.75
598.755.795.79
564.735.345.34
718.825.915.91
694.796.166.16
561.653.643.64
565.683.083.08
575.674.034.03
566.663.683.68
591.764.424.42
562.674.304.30
550.664.144.14
636.766.626.62
612.735.435.43
638.734.704.70
536.684.614.61
645.764.444.44
638.775.835.83