Assay Report Card

Basic Information

ID: ALA4670362

Type: Functional

Description: Antagonist activity at SNAP-tagged human GHSR expressed in HEK293 cells assessed as inhibition of ghrelin-induced IP1 accumulation at 10^-5M measured after 30 mins by IP1-d2 derivative based HTRF assay relative to ghrelin

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
508.633.963.96
665.805.505.50
603.734.674.67
656.765.975.97