Assay Report Card

Basic Information

ID: ALA4670371

Type: Functional

Description: Inverse agonist activity at SNAP-tagged human GHSR expressed in HEK293 cells assessed as inhibition of ghrelin-induced IP1 accumulation at 10^-5 M measured after 30 mins by HTRF assay relative to control

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
1347.66
902.153.813.81
677.816.036.03
688.834.834.83
706.855.795.79
702.826.216.21
725.855.205.20
732.856.216.21
656.795.465.46
707.846.126.12
669.815.795.79
652.765.055.05
693.815.735.73
700.844.984.98
642.765.075.07
679.785.435.43
672.793.813.81
688.793.523.52
707.846.126.12
681.775.865.86
715.863.883.88
685.834.704.70
663.785.725.72