ID: ALA4670371
Type: Functional
Description: Inverse agonist activity at SNAP-tagged human GHSR expressed in HEK293 cells assessed as inhibition of ghrelin-induced IP1 accumulation at 10^-5 M measured after 30 mins by HTRF assay relative to control
Organism: Homo sapiens
Cell type: HEK293
Bioactivity
Activity Types for Assay ALA4670371
Emax
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
1347.66 | ||
902.15 | 3.81 | 3.81 |
677.81 | 6.03 | 6.03 |
688.83 | 4.83 | 4.83 |
706.85 | 5.79 | 5.79 |
702.82 | 6.21 | 6.21 |
725.85 | 5.20 | 5.20 |
732.85 | 6.21 | 6.21 |
656.79 | 5.46 | 5.46 |
707.84 | 6.12 | 6.12 |
669.81 | 5.79 | 5.79 |
652.76 | 5.05 | 5.05 |
693.81 | 5.73 | 5.73 |
700.84 | 4.98 | 4.98 |
642.76 | 5.07 | 5.07 |
679.78 | 5.43 | 5.43 |
672.79 | 3.81 | 3.81 |
688.79 | 3.52 | 3.52 |
707.84 | 6.12 | 6.12 |
681.77 | 5.86 | 5.86 |
715.86 | 3.88 | 3.88 |
685.83 | 4.70 | 4.70 |
663.78 | 5.72 | 5.72 |