Basic Information
ID: ALA4670377
Type: Binding
Description: Inverse agonist activity at wild type human GHSR assembled into lipid nanodiscs assessed as reduction in ghrelin-induced decrease in proximity ratio at 10 uM after 30 mins by fluorophore-labelled TM1/TM6 probe-based FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4670377
Activity
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 732.85 | 6.21 | 6.21 |
| 693.81 | 5.73 | 5.73 |
| 679.78 | 5.43 | 5.43 |
| 663.78 | 5.72 | 5.72 |